A new butanolide compound from the aerial part of Lindera akoensis with anti-inflammatory activity.

نویسندگان

  • Chung-Ping Yang
  • Guan-Jhong Huang
  • Hui-Chi Huang
  • Yu-Chang Chen
  • Chi-I Chang
  • Sheng-Yang Wang
  • Ih-Sheng Chen
  • Yen-Hsueh Tseng
  • Shih-Chang Chien
  • Yueh-Hsiung Kuo
چکیده

A new butanolide, 3β-((E)-dodec-1-enyl)-4β-hydroxy-5β-methyldihydrofuran-2-one (1) and four known butanolides: Akolactone A (2), (3Z,4α,5β)-3-(dodec-11-enylidene)-4-hydroxy-5-methylbutalactone (3), (3E,4α,5β)-3-(dodec-11-enylidene)-4-hydroxy-5-methylbutalactone (4) and dihydroisoobtusilactone (5), were isolated from the aerial parts of Lindera akoensis. These butanolides showed in vitro anti-inflammatory activity decrease the LPS-stimulated production of nitrite in RAW264.7 cell, with IC₅₀ values of 1.4-179.9 μM.

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The Effect of the Aerial Part of Lindera akoensis on Lipopolysaccharides (LPS)-Induced Nitric Oxide Production in RAW264.7 Cells

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عنوان ژورنال:
  • Molecules

دوره 17 6  شماره 

صفحات  -

تاریخ انتشار 2012